Degarelix acetate is an antagonist of the gonadotropin-releasing hormone (GnRH) receptor, which is a synthetic substance. Its mechanism of action involves binding to the pituitary gland's GnRH receptor and inhibiting the release of gonadotropins and testosterone. As a result, it exerts an anti-prostate cancer effect.
Specifications
The chemical compound with the name Acetyl-(2S)-N-[(2S,3S)-3-{[(2S)-1-[(2R)-2-hydroxy-3-(naphthalen-2-yl)propanoyl]pyrrolidine-2-carbonyl]amino}-2-{3-[4-(2-hydroxyethyl)-1-piperazinyl]propyl}-3-methyl-L-valinamide is a complex structure consisting of several amino acids and compounds. It is commonly referred to as a peptide because of its composition.
The compound is formed by the combination of several amino acids, primarily valinamide, proline, and pyrrolidine-2-carbonyl. These amino acids provide the basis for the complex structure and the unique properties of the compound.
Acetyl-(2S)-N-[(2S,3S)-3-{[(2S)-1-[(2R)-2-hydroxy-3-(naphthalen-2-yl)propanoyl]pyrrolidine-2-carbonyl]amino}-2-{3-[4-(2-hydroxyethyl)-1-piperazinyl]propyl}-3-methyl-L-valinamide has several important applications in various fields, including pharmacology and biotechnology. Due to its complex composition, it can be used in a variety of different ways to achieve specific results.
Overall, Acetyl-(2S)-N-[(2S,3S)-3-{[(2S)-1-[(2R)-2-hydroxy-3-(naphthalen-2-yl)propanoyl]pyrrolidine-2-carbonyl]amino}-2-{3-[4-(2-hydroxyethyl)-1-piperazinyl]propyl}-3-methyl-L-valinamide is an important compound with diverse applications and unique properties. Its complex structure provides a unique advantage in various fields, and it continues to be a subject of research and development.
- Molecular Formula: C82H103ClN12O16
- Molecular Weight: 1632.44 g/mol
- CAS Number: 214766-78-6
- Purity ≥98%
- Impurity ≤0.5%
- Appearance: White to off-white powder
- Solubility: Soluble in water and methanol
Applications
Degarelix is an effective treatment for advanced prostate cancer as it acts as a receptor antagonist for gonadotropin-releasing hormone (GnRH). Its primary function is to decrease the testosterone level in the bloodstream, which proves beneficial in combating the progression of prostate cancer.
Why Use Degarelix Acetate：
Degarelix acetate is a potent medication prescribed for the management of advanced prostate cancer. By obstructing the production of cancer-stimulating hormones, it effectively hinders the growth and proliferation of cancer cells. This medication acts as a GnRH antagonist and is typically utilized when other hormone therapies fail to yield desired outcomes.
One notable advantage of degarelix is its rapid action in lowering testosterone levels. Consequently, this can result in a considerable reduction in both the size of the prostate and cancer activity. Administered through subcutaneous injections, degarelix acetate is generally well-tolerated and has minimal side effects.
Overall, degarelix acetate is an invaluable treatment option for men confronting the challenges posed by advanced prostate cancer. Its mechanism of action and effectiveness make it a crucial component in the fight against this disease, providing new hope for patients who have exhausted other treatment avenues.
Storage
- Keep the product in a cool and dry place with a temperature range of 20-25°C (68-77°F). It is essential to store it away from heat and direct sunlight.
- Protect from light and moisture.
- Keep out of reach of children.
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